Binding Binding Binding Binding Binding Binding AVP-induced cAMP inhibition AVP-induced cAMP inhibition AVP-induced cAMP inhibition AVP-induced cAMP inhibition AVP-induced cAMP inhibition AVP-induced cAMP inhibition
Ki nM Ki nM
Ratio Ki
pKi
SEM
n
Ki nM Ki nM Ratio Ki
pKi
SEM
n
MQ1 5.02 - 8.44 0.1 25 41 1 7,42 0,05 16
MQ2 8.16 1.6 8.17 0.15 4 98 2.4 7,04 0,1 3
MQ3 13.3 2.6 7.92 0.14 4 198 *** 4.8 6,71 0,07 3
MQ4 7.34 1.5 8.27 0.21 5 12 0.3 7,97 0,1 3
MQ5 3.50 0.7 8.58 0.3 4 9 0.2 8,17 0,3 5
MQ6 21.5 * 4.3 7.60 0.1 5 251 *** 6.1 6,66 0,2 3
MQ7-8 3.14 0.6 8.53 ND 2 25 0.6 7,65 0,2 3
MQ9 45.1 ** 9.0 7.35 ND 2 48 1.2 7,35 0,1 3
P19859 7.87 1.6 7.93 0.08 4 91 2.2 7,07 0,1 3
Q5ZPJ7 112 *** 112 *** 22.2 6.97 0.08 4 61 1.5 7,27 0,1 3
E7FL11 >>1000 >>1000 <<5 2 ND ND
B4ESA3 >>1000 >>1000 <<5 2 ND ND
C1IC51 >>1000 >>1000 <<5 2 ND ND
D5J9Q8 >>1000 >>1000 <<5 2 ND ND
F8J2F6 >>1000 >>1000 <<5 2 ND ND
D-DTx >>1000 >>1000 <<5 2 ND ND
DTx-K >>1000 >>1000 <<5 2 ND ND
α-DTx >>1000 >>1000 <<5 2 ND ND
DTx-I >>1000 >>1000 <<5 2 ND ND
Calci >>1000 >>1000 <<5 2 ND ND
BPTI >>1000 >>1000 <<5 2 ND ND